ADL-5859

SKU: orb1301009

Description

ADL-5859 hydrochloride is a potent and selective δ-opioid receptor agonist (Ki = 0.8 nM) with minimal activity at κ- and μ-opioid receptors and low hERG channel inhibition. It is a valuable research tool for investigating δ-receptor pharmacology in both in vitro assays and in vivo models of pain and mood disorders.

Research Area

Metabolism Research, Neuroscience, Pharmacology & Drug Discovery

Key Properties

• CAS Number: 850173-95-4
• MW: 428.95
• Purity: 98.78% (May vary between batches)
• Formula: C₂₄H₂₈N₂O₃·HCl
• SMILES: Cl.CCN(CC)C(=O)c1ccc(cc1)C1=CC2(CCNCC2)Oc2cccc(O)c12
• Target: Potassium Channel,Opioid Receptor,Cytochromes P450
• Solubility: DMSO:35 mg/mL (81.59 mM);Ethanol:1 mg/mL (2.33 mM);10% DMSO+40% PEG300+5% Tween-80+45% Saline:2 mg/mL (4.66 mM);H2O:5 mg/mL (11.66 mM)

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

ADL 5859, ADL 5859 Hydrochloride, ADL5859, ADL-5859, ADL-5859 Hydrochloride, Opioid Receptor, OpioidReceptor, δ-opioid receptor, μ-opioid receptor, κ-opioid receptor

Quick Database Links

Gene Symbol

Potassium Channel,Opioid Receptor,Cytochromes P450