AM1241

SKU: orb1300496

Description

AM-1241 is a potent and selective cannabinoid CB2 receptor agonist, demonstrating a Ki of 3.4 nM and 82-fold selectivity versus the CB1 receptor. It is widely used in preclinical research to investigate CB2 receptor function in models of pain, inflammation, and neuroprotection in both in vitro and in vivo studies.

Research Area

Pharmacology & Drug Discovery

Key Properties

• CAS Number: 444912-48-5
• MW: 503.33
• Purity: 98.72% (May vary between batches)
• Formula: C₂₂H₂₂IN₃O₃
• SMILES: C(=O)(C=1C=2C(N(CC3N(C)CCCC3)C1)=CC=CC2)C4=CC(N(=O)=O)=CC=C4I
• Target: Cannabinoid Receptor
• Solubility: Ethanol:< 1 mg/mL (insoluble or slightly soluble);10% DMSO + 40% PEG300 + 5% Tween 80 + 45% Saline:5 mg/mL (9.93 mM);H2O:< 1 mg/mL (insoluble or slightly soluble);DMSO:32.86 mg/mL (65.29 mM)

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

AM-1241, AM1241, AM 1241, CB2, CB1, Cannabinoid Receptor, CannabinoidReceptor

Quick Database Links

Gene Symbol

Cannabinoid Receptor