[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate

SKU: orb1296427

Description

[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate is a broad-spectrum neuropeptide antagonist and inverse agonist. It potently inhibits the ghrelin receptor and blocks tachykinin, bradykinin, CCK, and bombesin receptors. This compound has been shown to induce apoptosis and suppress cancer cell proliferation in vitro, making it a valuable tool for oncology and neuropharmacology research.

Research Area

Immunology & Inflammation, Pharmacology & Drug Discovery

Key Properties

• Target: Cholecystokinin Receptor
• MW: 1576.91
• Purity: 95.91% (May vary between batches)
• Formula: C₈₁H₁₁₃N₁₉O₁₄
• SMILES: CC(C)C[C@@H](C(N)=O)NC([C@H](CC(C)C)NC([C@@H](CC1=CNC2=C1C=CC=C2)NC([C@H](CC3=CC=CC=C3)NC([C@@H](CC4=CNC5=C4C=CC=C5)NC([C@H](CCC(N)=O)NC([C@@H](CC6=CC=CC=C6)NC([C@H]7N(C([C@H](CCCCN)NC([C@H]8N(C([C@@H](CCCNC(N)=N)N)=O)CCC8)=O)=O)CCC7)=O)=O)=O)=O)=O)=O)=O.CC(O)=O

Storage & Handling

• Storage: keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

CCK, [D Arg1,D Phe5,D Trp7,9,Leu11] Substance P acetate, [DArg1,DPhe5,DTrp7,9,Leu11]Substance P acetate, [D-Arg-1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate, [D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate(96736-12-8 free base)

Quick Database Links

Gene Symbol

Cholecystokinin Receptor