EED-226

SKU: orb1304185

Description

EED226 is a potent and selective small molecule inhibitor of the Embryonic Ectoderm Development (EED) protein, demonstrating an IC50 of 22 nM. Its oral bioavailability facilitates research into PRC2 function in both cellular assays and animal models for oncology and developmental biology studies.

Research Area

Epigenetics & Chromatin, Immunology & Inflammation

Key Properties

• CAS Number: 2083627-02-3
• MW: 369.40
• Purity: >98%
• Formula: C₁₇H₁₅N₅O₃S
• SMILES: N(CC1=CC=CO1)C=2N3C(C(=CN2)C4=CC=C(S(C)(=O)=O)C=C4)=NN=C3
• Target: Protein methyltransferase
• Solubility: Soluble in DMSO (up to 25 mg/ml)

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

antitumor, inhibit, K27me3, EED, EED-226, EED 226, EED226, HistoneMethyltransferase, Histone Methyltransferase, Inhibitor, PRC2

Quick Database Links

Gene Symbol

Protein methyltransferase