FLTX1

SKU: orb1298469

Description

FLTX1 is a fluorescent Tamoxifen analog that specifically labels intracellular estrogen receptors in both permeabilized and live cells. It functions as a pure antiestrogen, inhibiting estrogen receptor activity in breast cancer research models without uterine agonist effects, making it valuable for imaging and mechanistic studies.

Research Area

Metabolism Research

Key Properties

• CAS Number: 1481401-71-1
• MW: 520.58
• Purity: 98.42% (May vary between batches)
• Formula: C₃₁H₂₈N₄O₄
• SMILES: C(=C(/CC)\C1=CC=CC=C1)(\C2=CC=C(OCCN(C)C=3C=4C(C(N(=O)=O)=CC3)=NON4)C=C2)/C5=CC=CC=C5
• Target: Estrogen Receptor/ERR,Estrogen/progestogen Receptor
• Solubility: DMSO:5.21 mg/mL (10.01 mM)

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

FLTX1, FLTX 1, FLTX-1, ERR, fluorescent, ERα, Estrogen Receptor, estrogen, EstrogenReceptor, Estrogen Receptor/ERR, Inhibitor, inhibit, non-permeabilized, breast, antiestrogenic, cancer, progestogen Receptor, receptor, permeabilized, progestogenReceptor, Tamoxifen, uterus

Quick Database Links

Gene Symbol

Estrogen Receptor/ERR,Estrogen/progestogen Receptor