G-1

SKU: orb1308286

Description

G-1 is a nonsteroidal, high-affinity, and selective agonist for GPR30 (GPER), with a Ki value of 11 nM. This compound is employed in both in vitro and in vivo research to study GPER-mediated signaling in fields such as oncology, cardiology, endocrinology, and neuroscience, as documented in scientific literature.

Research Area

Metabolism Research, Pharmacology & Drug Discovery

Key Properties

• CAS Number: 881639-98-1
• MW: 412.28
• Purity: 98.14% (May vary between batches)
• Formula: C₂₁H₁₈BrNO₃
• SMILES: [H][C@@]12CC=C[C@]1([H])c1cc(ccc1N[C@@H]2c1cc2OCOc2cc1Br)C(C)=O
• Target: Estrogen Receptor/ERR,GPCR
• Solubility: DMSO:120 mg/mL (291.06 mM);H2O:< 0.1 mg/mL (insoluble);10% DMSO+40% PEG300+5% Tween 80+45% Saline:2 mg/mL (4.85 mM)

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

ERR, G 1, Estrogen Receptor/ERR, EstrogenReceptor, Estrogen Receptor, GPR30, G1, G-1, inhibit, Inhibitor

Quick Database Links

Gene Symbol

Estrogen Receptor/ERR,GPCR