GS-6201

SKU: orb1308258

Description

GS-6201 (CVT-6883) is a potent and selective adenosine A2B receptor antagonist with a Ki of 22 nM for the human receptor. This small molecule is a valuable research tool for investigating the role of A2B signaling in areas such as fibrosis, inflammation, and cancer in both cellular and animal models.

Research Area

Neuroscience, Pharmacology & Drug Discovery

Key Properties

• CAS Number: 752222-83-6
• MW: 446.43
• Purity: 98.32% (May vary between batches)
• Formula: C₂₁H₂₁F₃N₆O₂
• SMILES: CCCn1c(=O)n(CC)c2[nH]c(nc2c1=O)-c1cnn(Cc2cccc(c2)C(F)(F)F)c1
• Target: Adenosine Receptor
• Solubility: 10% DMSO+90% Corn Oil:2 mg/mL (4.48 mM);DMSO:30 mg/mL (67.2 mM)

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

human A1 receptors, human A2A receptors, human A2B receptors, human A3 receptors, GS6201, GS-6201, GS 6201, inhibit, Inhibitor, infarction, myocardial, caspase-1, cardiac, CVT 6883, CVT-6883, CVT6883, A2B, acute, airway, affinity, Adenosine Receptor, AdenosineReceptor, selectivity, P1 receptor, reactivity, remodeling

Quick Database Links

Gene Symbol

Adenosine Receptor