GSK1292263

SKU: orb1305147

Description

GSK1292263 is a selective agonist of the G-protein coupled receptor 119 (GPR119). It has been studied in preclinical research for its potential to stimulate glucose-dependent insulin secretion, making it a candidate for type 2 diabetes mellitus investigation in both in vitro and in vivo models.

Research Area

Metabolism Research, Pharmacology & Drug Discovery

Key Properties

• CAS Number: 1032823-75-8
• MW: 456.56
• Purity: 98.34% (May vary between batches)
• Formula: C₂₃H₂₈N₄O₄S
• SMILES: CC(C)c1noc(n1)N1CCC(COc2ccc(nc2)-c2ccc(cc2)S(C)(=O)=O)CC1
• Target: GPCR
• Solubility: Ethanol:< 1 mg/mL (insoluble or slightly soluble);DMSO:32 mg/mL (70.09 mM);10% DMSO+90% Corn Oil:2 mg/mL (4.38 mM)

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

GSK 1292263, GSK1292263, GSK-1292263, G Protein-Coupled Receptor 119, GPR119, Inhibitor, mellitus, inhibit, diabetes, T2DM, type

Quick Database Links

Gene Symbol

GPCR