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Istradefylline

SKU: orb1300666

Description

Istradefylline (KW-6002) is a potent and selective adenosine A2A receptor antagonist (Ki=2.2 nM) in Phase 3 development. Its research applications extend to Parkinson's disease, sleep disorders, and substance abuse, with studies utilizing both in vitro binding assays and in vivo models of neurological function.

Research Area

Neuroscience, Pharmacology & Drug Discovery

Images & Validation

Key Properties

CAS Number155270-99-8
MW384.43
Purity98.18% (May vary between batches)
FormulaC20H24N4O4
SMILESCN1C2=C(N(CC)C(=O)N(CC)C2=O)N=C1/C=C/C3=CC(OC)=C(OC)C=C3
TargetAdenosine Receptor
SolubilityDMSO:13.38 mg/mL (34.8 mM)

Storage & Handling

Storage-20°C
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

Alternative Names

Istradefylline, inhibit, KW6002, KW-6002, KW 6002, Inhibitor, P1 receptor, A2A, AdenosineReceptor, Adenosine Receptor

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  • Istradefylline [orb1226106]

    >98% (HPLC)

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    C20H24N4O4

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Istradefylline (orb1300666)

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Available Sizes

Select a size below

1 ml x 10 mM (in DMSO)
$ 80.00
5 mg
$ 80.00
10 mg
$ 90.00
25 mg
$ 120.00
50 mg
$ 140.00
100 mg
$ 190.00
500 mg
$ 420.00
DispatchUsually dispatched within 3-5 working days
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