Pitolisant hydrochloride

SKU: orb1300008

Description

Pitolisant hydrochloride, also known as Ciproxidine, is a highly potent and selective inverse agonist for the histamine H₃ receptor, exhibiting a Ki of 0.16 nM. It is widely used in neuroscience research, including in vitro binding assays and in vivo studies investigating sleep/wake disorders and cognitive functions.

Research Area

Immunology & Inflammation, Neuroscience, Pharmacology & Drug Discovery

Images & Validation

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Key Properties

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CAS Number	903576-44-3
MW	332.31
Purity	99.26% (May vary between batches)
Formula	C₁₇H₂₇Cl₂NO
SMILES	Cl.Clc1ccc(CCCOCCCN2CCCCC2)cc1
Target	Histamine Receptor
Solubility	DMSO:50 mg/mL (150.46 mM)

Storage & Handling

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Storage	-20°C
Expiration Date	12 months from date of receipt.
Disclaimer	For research use only

Alternative Names

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H3 receptor, Inhibitor, Histamine Receptor, HistamineReceptor, inhibit, Ciproxidine, BF 2649, BF2649, BF-2649, Pitolisant, Pitolisant hydrochloride, Pitolisant Hydrochloride

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Gene Symbol

Histamine Receptor

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