TC-G-1008

SKU: orb1302683

Description

TC-G-1008 (GPR39-C3) is a potent and selective agonist of the zinc-sensing receptor GPR39, demonstrating sub-nanomolar EC50 values for both human and rat orthologs. This compound is a valuable research tool for investigating GPR39's role in metabolic regulation, endocrine function, and neurological processes in both cellular and animal models.

Research Area

Pharmacology & Drug Discovery

Key Properties

• CAS Number: 1621175-65-2
• MW: 418.9
• Purity: 97.37% (May vary between batches)
• Formula: C₁₈H₁₉ClN₆O₂S
• SMILES: CNc1nc(NCc2ccc(NS(C)(=O)=O)cc2Cl)cc(n1)-c1ccccn1
• Target: GHSR
• Solubility: DMSO:255 mg/mL (608.74 mM);10% DMSO+40% PEG300+5% Tween 80+45% Saline:2 mg/mL (4.77 mM)

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

inhibit, Inhibitor, hGPR39, GPR39-C3, Growth hormone secretagogue receptor, GHSR, GHS-R, rGPR39, TC G 1008, TC-G 1008, TCG1008, TC-G1008, TC-G-1008

Quick Database Links

Gene Symbol

GHSR