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AM251

SKU: orb1225865

Description

AM251 is a potent CB1 receptor antagonist (IC50 = 8 nM, Ki = 7.49 nM) that displays 306-fold selectivity over CB2 receptors; also potent GPR55 agonist (EC50 = 39 nM).

Images & Validation

Key Properties

CAS Number183232-66-8
MW555.24
Purity>98% (HPLC)
FormulaC22H21Cl2IN4O
SMILESO=C(C1=NN(C2=CC=C(Cl)C=C2Cl)C(C3=CC=C(I)C=C3)=C1C)NN4CCCCC4
TargetCannabinoid Receptor
SolubilityDMSO: 40 mg/mL (72.04 mM)

Storage & Handling

StorageStorage temperature: -20°C. Stability: ≥ 2 years
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

Alternative Names

AM251 | AM 251 | AM-251

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  • AM251 [orb1307120]

    >98%

    183232-66-8

    555.24

    C22H21Cl2IN4O

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AM251 (orb1225865)

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200 mg
500 mg
5 mg
$ 90.00
10 mg
$ 130.00
25 mg
$ 220.00
50 mg
$ 380.00
100 mg
$ 550.00