Clobenpropit dihydrobromide

SKU: orb1298934

Description

Clobenpropit dihydrobromide is a potent histamine H3 receptor (H3R) antagonist and inverse agonist with a pEC50 of 8.07. This compound is widely used in neuroscience research to study H3R function in vitro and has been applied in vivo to explore its potential in models of cognitive disorders and sleep-wake regulation.

Research Area

Cell Biology, Immunology & Inflammation, Neuroscience, Pharmacology & Drug Discovery

Key Properties

• CAS Number: 145231-35-2
• MW: 470.7
• Purity: 99.48% (May vary between batches)
• Formula: C₁₄H₁₉Br₂ClN₄S
• SMILES: Br.Br.Clc1ccc(CNC(=N)SCCCc2cnc[nH]2)cc1
• Target: Apoptosis,Histamine Receptor
• Solubility: 10% DMSO+40% PEG300+5% Tween 80+45% Saline:1 mg/mL (2.12 mM);DMSO:4.71 mg/mL (10.01 mM)

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

Clobenpropit, Clobenpropit dihydrobromide, Clobenpropit Dihydrobromide, agonist, cancer, antagonist, Apoptosis, inhibit, inverse, pancreatic, HistamineReceptor, Histamine Receptor, histamine H3R, Inhibitor, H3 receptor, H3LR

Quick Database Links

Gene Symbol

Apoptosis,Histamine Receptor